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Tag Archives: PF-04457845
Discovery of PF-04457845 (FAAH Inhibitor)
In this latest publication from the Pfizer labs, the authors describe their continuing efforts to identify urea-based, irreversible inhibitors of fatty acid amide hydrolase (FAAH). Inhibition of FAAH and the concomitant elevation of endogenous levels of fatty acid amides has … Continue reading
Posted in Clinical Candidates, Enzyme Inhibitors
Tagged Analgesic, CYP450, FAAH, Fatty acid amide hydrolase, osteoarthritis, Pain, PF-04457845, PF-3845, Pfizer, Phase II, POC, PSA
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